Gestodene
13 -ethyl- 17β -hydroxy- 18 ,19- dinor -4 ,15- pregnadiene -20 -in- 3-one
G03AA10 G03AB06
Progestins
1.177 g · cm -1
197-198 ° C
Template: Infobox chemical / molecular formula search available
Gestodene is a synthetic progestin of the third generation, which is used as a hormonal contraceptive for birth control.
It is a selective, highly potent progestagen antigonadotrop. The antigonadotropic effect is about three times stronger than that of levonorgestrel. As the only progestagen it has a aldosteronantagonistischen effect, which is caused by a high affinity for the progesterone receptor. It also has minimal androgenic residual effect and a weak anti-estrogenic effect. Gestodene is exclusively in combination with ethinyl estradiol in the form of capsules and tablets on the market.
Trade names
Femovan (D), Minulet (D, A, CH), Minesse (A, CH), Mirelle (A, CH), tri- Minulet (FR)